SCHEMBL6233543

SCHEMBL6233543

Cc1c([N+](=O)[O-])ccc2sc(C(N)=O)c(C)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.40
TSHR P16473 5/20 0.39
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.38
CDC7 O00311 2/20 0.37
PLK4 O00444 2/20 0.37
DYRK3 O43781 2/20 0.37
ROCK2 O75116 2/20 0.37
PRKD3 O94806 2/20 0.37
MAP4K4 O95819 2/20 0.37
INSR P06213 2/20 0.37
CDK1 P06493 2/20 0.37
ROS1 P08922 2/20 0.37
PIM1 P11309 2/20 0.37
FGFR1 P11362 2/20 0.37
PRKACA P17612 2/20 0.37
RPS6KB1 P23443 2/20 0.37
CDK2 P24941 2/20 0.37
FLT4 P35916 2/20 0.37
KDR P35968 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11797546 0.75 TSHR (0.44) TDP1TSHRALDH1A1MAPTGAA
SCHEMBL2889156 0.71 TSHR (0.53) TDP1TSHRALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL5410548 0.70 LIMK1 (0.45) TSHRALDH1A1CDC7PLK4DYRK3
SCHEMBL5120287 0.70 TDP1 (0.46) TDP1TSHRALDH1A1MAPTSMN1; SMN2
SCHEMBL1117860 0.69 TSHR (0.50) TDP1TSHRALDH1A1MAPTSMN1; SMN2
SCHEMBL3828432 0.69 LIMK1 (0.47) TSHRALDH1A1MAPTCDC7PLK4
SCHEMBL30616318 0.67 TSHR (0.47) TDP1TSHRALDH1A1MAPTSMN1; SMN2
SCHEMBL28247578 0.67 L3MBTL1 (0.44) TDP1TSHRALDH1A1MAPTSMN1; SMN2
SCHEMBL7103494 0.67 TDP1 (0.39) TDP1TSHRALDH1A1MAPTSMN1; SMN2
SCHEMBL31440618 0.67 BCAT2 (0.39) ALDH1A1CDC7PLK4DYRK3ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed