SCHEMBL6233722

SCHEMBL6233722

Nc1nc(C(F)(F)F)c(-c2cccc(C(F)(F)F)c2)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 6/20 0.47
ADORA2A P29274 3/20 0.46
ADORA1 P30542 2/20 0.46
EPHX2 P34913 1/20 0.45
SCN4A P35499 1/20 0.45
XDH P47989 1/20 0.45
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
IKBKB O14920 1/20 0.43
BRD4 O60885 1/20 0.43
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CTSS P25774 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
LTA4H P09960 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL330359 0.84 BRD4 (0.51) RORBADORA2AADORA1EPHX2SCN4A
SCHEMBL332040 0.82 ALDH1A1 (0.58) ADORA2AADORA1MAPK1ALDH1A1SMN1; SMN2
SCHEMBL14364302 0.80 RORB (0.44) RORBADORA2AADORA1EPHX2SCN4A
SCHEMBL8237626 0.79 RORB (0.43) RORBADORA2AADORA1EPHX2SCN4A
SCHEMBL5048775 0.79 ALDH1A1 (0.52) RORBADORA2AADORA1XDHALDH1A1
SCHEMBL8708152 0.78 RORB (0.60) RORBADORA2AADORA1EPHX2SCN4A
SCHEMBL8240373 0.77 TGFBR1 (0.55) RORBADORA2AADORA1ALDH1A1CYP1A2
SCHEMBL27837167 0.76 ALDH1A1 (0.49) RORBADORA2AADORA1ALDH1A1SMN1; SMN2
SCHEMBL27837166 0.75 RORB (0.49) RORBADORA1XDHALDH1A1SMN1; SMN2
SCHEMBL923710 0.75 KDM4E (0.67) RORBALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed