SCHEMBL6234577

SCHEMBL6234577

COc1ccccc1C(C#N)(OC)OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
CA12 O43570 1/20 0.44
CA4 P22748 1/20 0.44
CA14 Q9ULX7 1/20 0.44
AR P10275 5/20 0.38
IMPDH2 P12268 1/20 0.38
IMPDH1 P20839 1/20 0.38
PGR P06401 1/20 0.38
ALDH1A1 P00352 4/20 0.38
TP53 P04637 1/20 0.38
TSHR P16473 1/20 0.38
ADRA2B P18089 1/20 0.38
PTGS1 P23219 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GAA P10253 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558441 0.78 CA1 (0.46) CA1CA2CA7CA9CA12
SCHEMBL31347528 0.78 CA1 (0.46) CA1CA2CA7CA9CA12
SCHEMBL30040149 0.77 AR (0.44) CA1CA2CA7CA9CA12
SCHEMBL14360010 0.77 AR (0.44) CA1CA2CA7CA9CA12
SCHEMBL10802674 0.74 ALDH1A1 (0.33) ARIMPDH2IMPDH1ALDH1A1MAPK1
SCHEMBL8784754 0.73 CA1 (0.55) CA1CA2CA7CA9CA12
SCHEMBL5675558 0.73 CA1 (0.55) CA1CA2CA7CA9CA12
SCHEMBL3671684 0.73 CA1 (0.55) CA1CA2CA7CA9CA12
SCHEMBL28453996 0.72 CA1 (0.39) CA1CA2CA7CA9CA12
SCHEMBL4160048 0.71 CYP2D6 (0.40) ALDH1A1TSHRGAAMAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1523556-A1 METHODS OF TREATING CONDITIONS ASSOCIATED WITH AN EDG-1 RECEPTOR SRI INTERNATIONAL (US) 2005-04-20 EP disclosed
WO-2004009816-A1 METHODS OF TREATING CONDITIONS ASSOCIATED WITH AN EDG-1 RECEPTOR CERETEK LLC (US) 2004-01-29 WO disclosed