SCHEMBL6558441

SCHEMBL6558441

COc1ccccc1C(C)(C)C#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA12 O43570 1/20 0.46
CA4 P22748 1/20 0.46
CA14 Q9ULX7 1/20 0.46
AR P10275 5/20 0.40
IMPDH2 P12268 1/20 0.39
IMPDH1 P20839 1/20 0.39
ALDH1A1 P00352 3/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
ADRA2B P18089 1/20 0.39
PTGS1 P23219 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CASR P41180 1/20 0.39
PGR P06401 1/20 0.39
SGMS2 Q8NHU3 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31347528 1.00 CA1 (0.46) CA1CA2CA7CA9CA12
SCHEMBL3531673 0.82 AR (0.39) CA1CA2CA7CA9CA12
SCHEMBL8763114 0.80 TSHR (0.39) CA2ARIMPDH2IMPDH1ALDH1A1
SCHEMBL12585665 0.79 RIPK1 (0.46) ARALDH1A1TSHRSGMS2MAPK1
SCHEMBL14360010 0.78 AR (0.44) CA1CA2CA7CA9CA12
SCHEMBL30040149 0.78 AR (0.44) CA1CA2CA7CA9CA12
SCHEMBL6234577 0.78 CA1 (0.44) CA1CA2CA7CA9CA12
SCHEMBL31445000 0.78 NR3C1 (0.47) PGR
SCHEMBL27939162 0.78 NR3C2 (0.41) ARPGRKDM4E
SCHEMBL1448547 0.78 TDP1 (0.46) ALDH1A1TP53TSHRPTGS1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101969773-B compounds and methods for reducing uric acid WELLSTAT THERAPEUTICS CORP. (US) 2015-08-19 CN disclosed
CN-102976928-B Compounds for reducing uric acid WELLSTAT THERAPEUTICS CORP 2014-09-17 CN disclosed
CN-101687773-B Substituted 2- [2- (phenyl) ethylamino ] alkanamide derivatives and their use as sodium and/or calcium channel modulators NEWRON PHARM SPA 2014-07-30 CN disclosed
CN-102976928-A Compounds for reducing uric acid WELLSTAT THERAPEUTICS CORP 2013-03-20 CN disclosed
CN-101687773-A Substituted 2- [ 2- (phenyl) ethylamino ] alkanamide derivatives and their use as sodium and/or calcium channel modulators NEWRON PHARM SPA 2010-03-31 CN disclosed
CN-101277939-A Acyclic ikur inhibitors BRISTOL MYERS SQUIBB CO (US) 2008-10-01 CN disclosed
CN-1768050-A Benzopyran compounds for the treatment of inflammation PHARMACIA CORP (US) 2006-05-03 CN disclosed
CN-1250528-C Cyclic nitrones and pharmaceutical compositions containing them AWENTIS PHARMACEUTICAL INC (US) 2006-04-12 CN disclosed
EP-1046635-B1 Process for preparing an aromatic compound substituted by a tertiary nitrile PFIZER PROD INC (US) 2004-12-29 EP disclosed
CN-1500787-A Cyclic nitrones and pharmaceutical compositions containing them ���µ�˹ҩ�﹫˾ 2004-06-02 CN disclosed
CN-1500779-A Cyclic nitrones and pharmaceutical compositions containing them ���µ�˹ҩ�﹫˾ 2004-06-02 CN disclosed
US-6358974-B1 USED AS AS MODULATORS OF DOPAMINE D.SUB.3 RECEPTORS, IN THERAPY AS ANTIPSYCHOTIC AGENTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-03-19 US disclosed
US-6303782-B1 TREATING A FLUORINE-SUBSTITUTED AROMATIC COMPOUND WITH A SECONDARY NITRILE IN THE PRESENCE OF A BASE PFIZER INC 2001-10-16 US disclosed
EP-1137638-A2 ISOQUINOLINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2001-10-04 EP disclosed
EP-1046635-A1 Process for preparing an aromatic compound substituted by a tertiary nitrile Pfizer Products Inc. (US) 2000-10-25 EP disclosed
WO-2000024717-A2 ISOQUINOLINE DERIVATIVES SMITHKLINE BEECHAM P.L.C. (GB) 2000-05-04 WO disclosed
CN-1196050-A Cyclic nitrones and pharmaceutical compositions containing them HOECHST MARION ROUSSEL INC (US) 1998-10-14 CN disclosed
US-4333759-A Herbicidal 5-cyano-2,3-dihydro-benzofuran-2-ones FISONS LIMITED (GB) 1982-06-08 US disclosed
US-4263037-A 5-Cyano-2,3-dihydrobenzofurans useful as herbicides FISONS LIMITED (GB) 1981-04-21 US disclosed
EP-0007719-A2 Cyanbenzofuran derivatives, processes for their preparation and their use in herbicidal compositions; cyanobenzene, benzodioxepine, benzodioxaphosphepine and benzodioxathiepine derivatives FBC LIMITED (GB) 1980-02-06 EP disclosed