SCHEMBL6234629

SCHEMBL6234629

COc1ccc(Nc2nc(N)nc(NCC3CCCN3C)n2)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GALR1 P47211 7/20 0.48
GALR2 O43603 6/20 0.47
CDK1 P06493 1/20 0.41
CDK4 P11802 1/20 0.41
CCNB1 P14635 1/20 0.41
CCND1 P24385 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CAMK2D Q13557 1/20 0.40
DHFR P00374 1/20 0.40
EPHA2 P29317 1/20 0.39
KDR P35968 1/20 0.39
EPHB4 P54760 1/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5036029 0.90 GALR1 (0.61) GALR1GALR2CDK1CDK4CCNB1
SCHEMBL5551996 0.89 GALR1 (0.47) GALR1GALR2MAPT
SCHEMBL5553433 0.88 GALR1 (0.50) GALR1GALR2CDK1CDK4CCNB1
SCHEMBL4829744 0.83 DRD2 (0.50) GALR1GALR2
SCHEMBL4832495 0.83 DRD2 (0.50) GALR1GALR2
SCHEMBL4838923 0.83 GALR1 (0.67) GALR1GALR2CDK1CDK4CCNB1
SCHEMBL4836437 0.81 GALR1 (0.48) GALR1GALR2
SCHEMBL5031357 0.80 GALR1 (0.54) GALR1GALR2
SCHEMBL4832704 0.80 GALR1 (0.50) GALR1GALR2MAPTMAPK1TDP1
SCHEMBL6921463 0.80 KCNH3 (0.60) GALR1USP2ALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1560817-A1 METHODS AND COMPOSITIONS OF NOVEL TRIAZINE COMPOUNDS Reddy US Therapeutics, Inc. (US) 2005-08-10 EP claimed
WO-2004026844-A9 METHODS AND COMPOSITIONS OF NOVEL TRIAZINE COMPOUNDS REDDY US THERAPEUTICS INC (US) 2004-11-11 WO claimed
WO-2004026844-A1 METHODS AND COMPOSITIONS OF NOVEL TRIAZINE COMPOUNDS REDDY US THERAPEUTICS, INC. (US) 2004-04-01 WO claimed