SCHEMBL6235619

SCHEMBL6235619

CCCC(C(=O)O)C(O)CBr

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.44
CHRM1 P11229 1/20 0.44
AKR1A1 P14550 1/20 0.44
CHRM3 P20309 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
ADRA1A P35348 1/20 0.44
HRH1 P35367 1/20 0.44
DRD3 P35462 1/20 0.44
SLC6A3 Q01959 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
GPR84 Q9NQS5 5/20 0.38
FFAR1 O14842 1/20 0.38
LCK P06239 1/20 0.36
PPARD Q03181 1/20 0.36
ZDHHC20 Q5W0Z9 1/20 0.36
ZDHHC2 Q9UIJ5 1/20 0.36
TSHR P16473 3/20 0.36
ALDH1A1 P00352 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10780881 1.00 TDP1 (0.44) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL6243346 0.88 CA2 (0.45) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL10774519 0.84 GPR84 (0.55) GPR84FFAR1LCKPPARDZDHHC20
SCHEMBL10774525 0.84 GPR84 (0.55) GPR84FFAR1LCKPPARDZDHHC20
SCHEMBL676549 0.84 TDP1 (0.50) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL9636422 0.82 TDP1 (0.48) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL10774556 0.82 ALDH1A1 (0.39) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL13986496 0.82 TDP1 (0.48) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL1000793 0.82 TDP1 (0.48) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL606891 0.82 ALDH1A1 (0.39) TDP1CHRM1AKR1A1CHRM3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005375-A1 METHOD FOR PRODUCING 4-CYANO-3-HYDROXYBUTYRIC ACID ESTERS LANXESS DEUTSCHLAND GMBH (DE) 2005-01-20 WO claimed
WO-2005005375-A1 METHOD FOR PRODUCING 4-CYANO-3-HYDROXYBUTYRIC ACID ESTERS LANXESS DEUTSCHLAND GMBH (DE) 2005-01-20 WO disclosed