SCHEMBL6236296

SCHEMBL6236296

COC(=O)c1ccc(Cc2cc3c(cc2OC)C(C)(C)CCC3(C)C)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 8/20 0.55
CYP3A4 P08684 4/20 0.52
RXRB P28702 1/20 0.49
RXRG P48443 1/20 0.49
CYP26A1 O43174 2/20 0.48
FPR1 P21462 1/20 0.45
GNRHR P30968 1/20 0.45
GPR183 P32249 1/20 0.45
GPR119 Q8TDV5 1/20 0.45
HNF4A P41235 2/20 0.44
KMT2A Q03164 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.42
RARA P10276 1/20 0.42
RARB P10826 1/20 0.42
RARG P13631 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MAPT P10636 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6238178 0.89 RXRA (0.56) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6244434 0.89 RXRA (0.70) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6240226 0.88 RXRA (0.51) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6245896 0.87 RXRA (0.51) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6237264 0.87 RXRA (0.51) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6903012 0.86 RXRA (0.74) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6241202 0.86 RXRA (0.56) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6242960 0.84 RXRA (0.47) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL6238864 0.84 RXRA (0.48) RXRACYP3A4RXRBRXRGCYP26A1
SCHEMBL8016720 0.79 CYP3A4 (0.56) RXRACYP3A4RXRBRXRGCYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005017185-A2 HEPATOCYTE NUCLEAR FACTOR 4α MODULATOR COMPOUNDS LIGAND PHARMCEUTICALS INCORPORATED (US) 2005-02-24 WO disclosed