SCHEMBL6237061

SCHEMBL6237061

O=Cc1cnc2[nH]cncc1-2

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.31
FKBP5 Q13451 1/20 0.31
CCNT1 O60563 1/20 0.31
CDK9 P50750 1/20 0.31
HASPIN Q8TF76 1/20 0.31
MEN1 O00255 1/20 0.31
KDM4E B2RXH2 1/20 0.31
BLM P54132 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28071244 0.78 CCNT1 (0.33) CCNT1CDK9HASPIN
SCHEMBL18341916 0.71 ALDH1A1 (0.36) KMT2AALDH1A1FKBP5MEN1KDM4E
SCHEMBL25861866 0.69 ALDH1A1 (0.44) ALDH1A1FKBP5CYP3A4TSHR
SCHEMBL6502793 0.69 IDO1 (0.38) ALDH1A1FKBP5TSHR
SCHEMBL311677 0.69 ALDH1A1 (0.34) ALDH1A1FKBP5KDM4ENPSR1
SCHEMBL13725534 0.69 KMT2A (0.33) KMT2AALDH1A1FKBP5MEN1KDM4E
SCHEMBL21713005 0.68 CYP3A4 (0.39) KMT2AALDH1A1KDM4EBLMNPSR1
SCHEMBL28202370 0.67 ALDH1A1 (0.35) KMT2AALDH1A1MEN1KDM4ECYP3A4
SCHEMBL30200923 0.65 IDO1 (0.39) KDM4EBLMNPSR1CYP3A4TSHR
Hydrochloric Acid SCHEMBL28274257 0.64 HRH3 (0.33) ALDH1A1FKBP5KDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115838370-A EGFR inhibitor and preparation method and application thereof 山东新时代药业有限公司 2023-03-24 CN disclosed
EP-0836613-B1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS METABASIS THERAPEUTICS INC (US) 2005-05-25 EP disclosed
EP-0832092-B1 ORALLY ACTIVE ADENOSINE KINASE INHIBITORS METABASIS THERAPEUTICS INC (US) 2004-11-17 EP disclosed
EP-0836613-A1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-22 EP disclosed
EP-0832092-A1 ORALLY ACTIVE ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040706-A1 ORALLY ACTIVE ADENOSINE KINASE INHIBITORS GENSIA-SICOR (US) 1996-12-19 WO disclosed
WO-1996040707-A1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed