SCHEMBL6238622

SCHEMBL6238622

O=C(O)/C=C/c1ccc(Sc2ccc(F)cc2)c(Cl)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLA2G4A P47712 1/20 0.43
PTGES O14684 1/20 0.43
ITGB2 P05107 8/20 0.42
ICAM1 P05362 8/20 0.42
ITGAL P20701 8/20 0.42
MIF P14174 1/20 0.40
RHEB Q15382 1/20 0.40
TDO2 P48775 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
AGBL2 Q5U5Z8 1/20 0.37
KDM4E B2RXH2 2/20 0.36
HTT P42858 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6238628 1.00 PLA2G4A (0.43) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL6817329 0.85 ITGB2 (0.52) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL6568833 0.85 ITGB2 (0.52) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL6759499 0.81 PLA2G4A (0.54) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL6759492 0.81 PLA2G4A (0.54) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL4278689 0.79 MIF (0.44) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL4278685 0.79 MIF (0.44) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL4277853 0.76 PTGES (0.45) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL4277854 0.76 PTGES (0.45) PLA2G4APTGESITGB2ICAM1ITGAL
SCHEMBL6316878 0.76 ITGB2 (0.43) PLA2G4APTGESITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019177-A1 AMINOPIPERIDINE AMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed