SCHEMBL6239006

SCHEMBL6239006

NC(=O)[C@@H]1C[C@H](OCc2ccc(Cl)cc2)CN1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
CARM1 Q86X55 1/20 0.37
PRMT6 Q96LA8 1/20 0.37
GRM2 Q14416 1/20 0.37
GRM3 Q14832 1/20 0.37
IDO1 P14902 2/20 0.37
AGXT P21549 2/20 0.37
KCNH2 Q12809 2/20 0.36
HRH3 Q9Y5N1 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236176 1.00 EPHX2 (0.38) EPHX2NPC1RAB9AKMT2ACARM1
SCHEMBL8177812 0.88 GRIK1 (0.44) GRM2GRM3CYP2C9CYP2C19ALDH1A1
SCHEMBL3182056 0.88 GRIK1 (0.44) GRM2GRM3CYP2C9CYP2C19ALDH1A1
SCHEMBL30471875 0.86 KCNH2 (0.46) NPC1RAB9ACARM1PRMT6IDO1
SCHEMBL24928604 0.86 KCNH2 (0.44) EPHX2KCNH2CYP2C19ALDH1A1
SCHEMBL7385029 0.86 KCNH2 (0.44) EPHX2KCNH2CYP2C19ALDH1A1
SCHEMBL6238616 0.86 KCNH2 (0.44) EPHX2KCNH2CYP2C19ALDH1A1
SCHEMBL8151501 0.84 P2RX3 (0.48) EPHX2CARM1PRMT6ALDH1A1CYP3A4
SCHEMBL6239011 0.76 IDO1 (0.40) CARM1PRMT6IDO1AGXTSLC6A4
SCHEMBL6236177 0.76 IDO1 (0.40) CARM1PRMT6IDO1AGXTSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011697-A2 SULFONAMIDE DERIVATIVES WITH ACTIVITY ON PROTEIN KINASE A AND B ASTEX THERAPEUTICS LIMITED (GB) 2005-02-10 WO disclosed