SCHEMBL6239108

SCHEMBL6239108

O=[N+]([O-])c1[c]ccc(-c2cccc(Cl)c2Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSD A5PKW4 1/20 0.34
TDP1 Q9NUW8 3/20 0.34
ALDH1A1 P00352 3/20 0.33
SCN9A Q15858 1/20 0.33
PTGES2 Q9H7Z7 1/20 0.33
NOTUM Q6P988 1/20 0.33
BCL2L1 Q07817 1/20 0.33
MCL1 Q07820 1/20 0.33
CNR2 P34972 1/20 0.33
TSHR P16473 1/20 0.33
PDPK1 O15530 1/20 0.32
DHODH Q02127 1/20 0.32
MAPT P10636 2/20 0.32
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSP90AA1 P07900 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
USP7 Q93009 1/20 0.31
USP47 Q96K76 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1746866 0.88 CYP2A6 (0.40) TDP1ALDH1A1MAPTPOLBMEN1
SCHEMBL6190813 0.78 CNR2 (0.39) PSDTDP1ALDH1A1SCN9ANOTUM
SCHEMBL6192327 0.77 ALDH1A1 (0.47) TDP1ALDH1A1NOTUMTSHRMAPT
SCHEMBL6195275 0.77 ALDH1A1 (0.56) TDP1ALDH1A1MAPTMEN1HPGD
SCHEMBL15636896 0.76 CNR2 (0.41) SCN9APTGES2NOTUMCNR2TSHR
SCHEMBL6193171 0.76 PTPRC (0.41) TDP1ALDH1A1MAPTPOLB
SCHEMBL6194132 0.76 MCL1 (0.41) TDP1ALDH1A1MCL1TSHRCA1
SCHEMBL6190538 0.75 TDP1 (0.50) TDP1ALDH1A1TSHRDHODHMAPT
SCHEMBL6187317 0.75 AHR (0.47) TDP1NOTUMTSHRMAPTPOLB
SCHEMBL6232173 0.74 ALDH1A1 (0.38) TDP1ALDH1A1TSHRMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1585727-A1 INDOLES USEFUL IN THE TREATMENT OF ANDROGEN-RECEPTOR RELATED DISEASES Akzo Nobel N.V. (NL) 2005-10-19 EP disclosed
WO-2004041782-A1 INDOLES USEFUL IN THE TREATMENT OF ANDROGEN-RECEPTOR RELATED DISEASES AKZO NOBEL N.V. (NL) 2004-05-21 WO disclosed