SCHEMBL6232173

SCHEMBL6232173

O=[N+]([O-])c1[c]ccc(-c2cc(Cl)cc(Cl)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
TSHR P16473 3/20 0.38
TDP1 Q9NUW8 2/20 0.35
MAPK1 P28482 1/20 0.35
RXRA P19793 2/20 0.35
RXRB P28702 2/20 0.35
CYP19A1 P11511 1/20 0.33
HSD17B10 Q99714 1/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
TTR P02766 1/20 0.31
PGR P06401 1/20 0.31
VCAM1 P19320 1/20 0.31
KIF18A Q8NI77 1/20 0.30
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6192327 0.88 ALDH1A1 (0.47) ALDH1A1TSHRTDP1MAPK1RXRA
SCHEMBL6191703 0.88 AHR (0.38) ALDH1A1TSHRTDP1MAPK1CYP19A1
SCHEMBL6187317 0.83 AHR (0.47) TSHRTDP1MAPK1HSD17B10MEN1
SCHEMBL8650141 0.81 CYP19A1 (0.35) TSHRTDP1CYP19A1MEN1POLB
SCHEMBL387257 0.81 ALDH1A1 (0.44) ALDH1A1TSHRTDP1MAPK1HSD17B10
SCHEMBL3296222 0.80 CRHBP (0.49) ALDH1A1TDP1MAPK1CYP19A1POLB
SCHEMBL6191442 0.79 PGR (0.37) ALDH1A1TDP1CYP19A1MEN1POLB
SCHEMBL9206594 0.79 CA12 (0.44) ALDH1A1TDP1MAPK1CYP19A1HSD17B10
SCHEMBL5631988 0.77 HPRT1 (0.47) ALDH1A1TSHRTDP1MAPK1HSD17B10
SCHEMBL15208829 0.77 POLB (0.34) ALDH1A1TDP1CYP19A1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1585727-A1 INDOLES USEFUL IN THE TREATMENT OF ANDROGEN-RECEPTOR RELATED DISEASES Akzo Nobel N.V. (NL) 2005-10-19 EP disclosed
WO-2004041782-A1 INDOLES USEFUL IN THE TREATMENT OF ANDROGEN-RECEPTOR RELATED DISEASES AKZO NOBEL N.V. (NL) 2004-05-21 WO disclosed