SCHEMBL6239398

SCHEMBL6239398

C#Cc1cncc(OC(C)[C@@H]2CCCN2)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 9/20 0.43
CHRNA3 P32297 5/20 0.43
CHRNA4 P43681 8/20 0.37
CHRNB4 P30926 4/20 0.37
CHRNA1 P02708 3/20 0.37
CHRNG P07510 1/20 0.37
CHRNB1 P11230 1/20 0.37
CHRND Q07001 1/20 0.37
CHRNA2 Q15822 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4727579 1.00 CHRNB2 (0.43) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA1
SCHEMBL8550383 0.89 GPR119 (0.37) CHRNB2CHRNA3CHRNA4CHRNB4
SCHEMBL4727403 0.85 CHRNB2 (0.48) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA2
SCHEMBL6235429 0.83 CHRNB2 (0.54) CHRNB2CHRNA3CHRNA4CHRNB4CHRNB1
SCHEMBL8554594 0.82 CHRNB2 (0.41) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA2
SCHEMBL8553258 0.82 CHRNB2 (0.41) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA2
SCHEMBL6231934 0.82 CHRNB2 (0.48) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA2
SCHEMBL4726517 0.82 CHRNB2 (0.48) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA2
SCHEMBL7406929 0.81 CHRNB4 (0.36) CHRNB2CHRNA3CHRNA4CHRNB4
SCHEMBL4962971 0.81 CHRNB2 (0.49) CHRNB2CHRNA3CHRNA4CHRNB4CHRNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000806-A2 LIGANDS FOR NICOTINIC ACETYLCHOLINE RECEPTORS, AND METHODS OF MAKING AND USING THEM GEORGETOWN UNIVERSITY (US) 2005-01-06 WO disclosed