SCHEMBL6239581

SCHEMBL6239581

O=[N+]([O-])c1ccc2nc(Nc3cccc(F)c3)c(-c3cccs3)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 10/20 0.54
EGFR P00533 1/20 0.53
RHOA P61586 1/20 0.48
GUCY1B2 O75343 1/20 0.47
GUCY1A2 P33402 1/20 0.47
GUCY1A1 Q02108 1/20 0.47
GUCY1B1 Q02153 1/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 2/20 0.46
PIN1 Q13526 1/20 0.46
CYP1A2 P05177 2/20 0.43
AURKB Q96GD4 1/20 0.43
HCRTR1 O43613 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237490 0.84 ABCG2 (0.67) ABCG2EGFRMEN1KMT2AMAPT
SCHEMBL6232602 0.83 ABCG2 (0.55) ABCG2EGFRMEN1KMT2AMAPT
SCHEMBL7691382 0.82 ABCG2 (0.61) ABCG2EGFRMEN1KMT2AMAPT
SCHEMBL6237367 0.76 CYP1A2 (0.51) ABCG2GUCY1B2GUCY1A2GUCY1A1GUCY1B1
SCHEMBL17597920 0.74 GUCY1B2 (0.73) ABCG2EGFRRHOAGUCY1B2GUCY1A2
SCHEMBL19129480 0.72 GUCY1B2 (0.77) ABCG2EGFRRHOAGUCY1B2GUCY1A2
SCHEMBL7697772 0.72 RPS6KB2 (0.58) ABCG2MEN1KMT2AMAPTALDH1A1
SCHEMBL17598175 0.71 GUCY1B2 (0.76) ABCG2EGFRRHOAGUCY1B2GUCY1A2
SCHEMBL20299204 0.71 ABCG2 (0.72) ABCG2EGFRMEN1KMT2AMAPT
SCHEMBL22860661 0.71 EGFR (0.67) ABCG2EGFRRHOAGUCY1B2GUCY1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007099-A2 PKB INHIBITORS AS ANTI-TUMOR AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2005-01-27 WO disclosed