SCHEMBL6237490

SCHEMBL6237490

Fc1cccc(Nc2nc3ccccc3nc2-c2cccs2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 8/20 0.67
PDE5A O76074 1/20 0.49
AURKB Q96GD4 1/20 0.48
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
ABCB1 P08183 2/20 0.48
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 3/20 0.47
LMNA P02545 2/20 0.47
HPGD P15428 2/20 0.47
MAPT P10636 2/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
POLB P06746 1/20 0.47
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
RAB9A P51151 1/20 0.47
EGFR P00533 1/20 0.47
LCK P06239 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7691382 0.93 ABCG2 (0.61) ABCG2PDE5AAURKBKMT2AMEN1
SCHEMBL6232602 0.89 ABCG2 (0.55) ABCG2PDE5AAURKBKMT2AMEN1
SCHEMBL6259663 0.85 PDE5A (0.61) ABCG2PDE5AKMT2AMEN1ABCB1
SCHEMBL6235369 0.85 MEN1 (0.58) ABCG2PDE5AKMT2AMEN1ABCB1
SCHEMBL6236522 0.85 ABCG2 (0.48) ABCG2PDE5AKMT2AMEN1ABCB1
SCHEMBL6239609 0.84 MAPT (0.51) ABCG2PDE5AKMT2AMEN1ABCB1
SCHEMBL6239581 0.84 ABCG2 (0.54) ABCG2AURKBKMT2AMEN1ALDH1A1
SCHEMBL6239843 0.81 ABCG2 (0.53) ABCG2PDE5AKMT2AMEN1ABCB1
SCHEMBL7697772 0.79 RPS6KB2 (0.58) ABCG2PDE5AKMT2AMEN1ABCB1
SCHEMBL7697783 0.78 RPS6KB2 (0.57) ABCG2PDE5AKMT2AMEN1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007099-A2 PKB INHIBITORS AS ANTI-TUMOR AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2005-01-27 WO disclosed