SCHEMBL6239746

SCHEMBL6239746

Cc1cccc(C)c1N(C(N)=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 6/20 0.42
MEN1 O00255 1/20 0.42
CRHBP P24387 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
CRHR2 Q13324 1/20 0.42
TLR9 Q9NR96 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GAA P10253 2/20 0.41
NOS1 P29475 4/20 0.41
ACHE P22303 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LMNA P02545 1/20 0.41
AR P10275 1/20 0.40
TDP1 Q9NUW8 3/20 0.40
NOS3 P29474 2/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28425336 0.84 NPC1 (0.45) TSHRNPC1RAB9AALDH1A1MEN1
SCHEMBL1177204 0.82 TSHR (0.57) TSHRALDH1A1MEN1CRHBPKMT2A
SCHEMBL6037591 0.81 ESR1 (0.41) TSHRALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL7493116 0.80 RORC (0.43) TSHRNPC1RAB9AALDH1A1KMT2A
SCHEMBL11291473 0.80 ALDH1A1 (0.62) TSHRNPC1RAB9AALDH1A1MEN1
SCHEMBL28100013 0.79 ALDH1A1 (0.54) TSHRALDH1A1MEN1KMT2AGAA
SCHEMBL6792424 0.75 TSHR (0.49) TSHRALDH1A1MEN1CRHBPKMT2A
SCHEMBL4162102 0.74 TSHR (0.55) TSHRALDH1A1MEN1CRHBPKMT2A
SCHEMBL6037517 0.73 ESR1 (0.41) NPC1RAB9AALDH1A1ATMHSD17B10
SCHEMBL15659596 0.73 TSHR (0.53) TSHRALDH1A1MEN1CRHBPKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005021721-A2 CARBOXYLESTERASE INHIBITORS ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2005-03-10 WO claimed