SCHEMBL6242590

SCHEMBL6242590

COCCNS(=O)(=O)c1ccc(Nc2nccc(-c3c(C)nc4cccnn34)n2)cc1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 16/20 0.71
CDK4 P11802 8/20 0.61
CDK1 P06493 3/20 0.60
IKBKB O14920 3/20 0.45
CCNE1 P24864 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6243791 0.85 CDK2 (0.57) CDK2CDK4CDK1IKBKBCCNE1
SCHEMBL6244692 0.85 CDK2 (0.78) CDK2CDK4CDK1IKBKB
SCHEMBL6594955 0.83 CDK2 (1.00) CDK2CDK4CDK1IKBKB
SCHEMBL4820462 0.81 CDK2 (0.80) CDK2CDK4CDK1IKBKB
SCHEMBL4817036 0.81 CDK2 (0.79) CDK2CDK4CDK1IKBKBCCNE1
SCHEMBL6245840 0.80 CDK2 (0.76) CDK2CDK4CDK1IKBKB
SCHEMBL4821591 0.80 CDK2 (0.72) CDK2CDK4CDK1IKBKB
SCHEMBL7978102 0.78 CDK2 (0.50) CDK2CDK4CDK1CCNE1
SCHEMBL6245628 0.78 CDK2 (0.69) CDK2CDK4CDK1CCNE1
SCHEMBL4855523 0.78 CDK2 (0.83) CDK2CDK4CDK1IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362050-B1 PYRIMIDINE DERIVATIVES FOR INHIBITION OF CELL-PROLIFERATION ASTRAZENECA AB (SE) 2005-02-02 EP claimed