SCHEMBL624629

SCHEMBL624629

CCCc1ccc(C#Cc2cccnc2N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 13/20 0.47
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
CHRM2 P08172 1/20 0.39
S1PR1 P21453 1/20 0.39
FPR1 P21462 1/20 0.39
FPR3 P25089 1/20 0.39
GPR183 P32249 1/20 0.39
APLNR P35414 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
GPR65 Q8IYL9 1/20 0.39
NPC1 O15118 1/20 0.39
CASP3 P42574 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SENP8 Q96LD8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30270431 0.78 KDM4E (0.59) FFAR1ALDH1A1HPGDKDM4ECHRM2
SCHEMBL18952028 0.77 MAPT (0.57) FFAR1ALDH1A1HPGDKDM4ENPC1
SCHEMBL623035 0.76 ADK (0.45) FFAR1ALDH1A1HPGDL3MBTL1KDM4E
SCHEMBL8141107 0.75 ACACB (0.54) FFAR1FFAR4ACACB
SCHEMBL9328434 0.75 ACACB (0.54) FFAR1FFAR4ACACB
SCHEMBL9511319 0.73 ACACB (0.53) FFAR1FFAR4ACACB
SCHEMBL8455468 0.73 FFAR1 (0.68) FFAR1L3MBTL1CHRM2S1PR1FPR1
SCHEMBL29856280 0.73 NOS2 (0.44) ALDH1A1HPGDKDM4EGAANPC1
SCHEMBL12474028 0.72 MKNK1 (0.51) ALDH1A1HPGDKDM4EGAAFFAR4
SCHEMBL2833040 0.71 FFAR1 (0.58) FFAR1CHRM2S1PR1FPR1FPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2603513-A1 HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2013-06-19 EP disclosed
WO-2012020848-A1 HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-02-16 WO disclosed