SCHEMBL6246702

SCHEMBL6246702

NC(=O)C(C(N)=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.57
CES2 O00748 2/20 0.57
EPHX1 P07099 8/20 0.54
ACP3 P15309 1/20 0.53
IDO1 P14902 1/20 0.50
TDO2 P48775 1/20 0.50
TRPM8 Q7Z2W7 1/20 0.49
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
HTR3A P46098 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11431980 0.87 CES2 (0.49) PNMTCES2EPHX1ACP3TRPM8
SCHEMBL27890286 0.87 ALDH1A1 (0.50) PNMTCES2EPHX1ACP3IDO1
SCHEMBL8234510 0.86 PNMT (0.54) PNMTCES2EPHX1ACP3IDO1
SCHEMBL29658610 0.86 CES2 (0.67) PNMTCES2EPHX1ACP3IDO1
SCHEMBL5527951 0.86 CES2 (0.67) PNMTCES2EPHX1ACP3IDO1
SCHEMBL27996637 0.86 PNMT (0.54) PNMTCES2EPHX1ACP3IDO1
SCHEMBL18952889 0.85 CES2 (0.57) PNMTCES2EPHX1ACP3IDO1
SCHEMBL7469419 0.84 PNMT (0.53) PNMTCES2EPHX1ACP3IDO1
SCHEMBL377074 0.84 AURKA (0.57) PNMTCES2EPHX1ACP3
Hydrochloric Acid SCHEMBL28755205 0.84 PNMT (0.53) PNMTCES2EPHX1ACP3IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037196-A2 SUBSTITUTED 2-ARYLMETHYLENE-N-ARYL-N'-ARYL-MALONAMIDES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS CYTOVIA, INC. (US) 2005-04-28 WO claimed
CN-108026027-B Substituted malonamide compounds and their use as antibacterial agents 邱浩杰 2020-10-02 CN disclosed
WO-2020039601-A1 OIL-IN-WATER TYPE EMULSION OF ACTINIC-RAY-CURABLE RESIN COMPOSITION, AND THERMAL RECORDING MATERIAL 日本化薬株式会社 2020-02-27 WO disclosed
WO-2005037196-A2 SUBSTITUTED 2-ARYLMETHYLENE-N-ARYL-N'-ARYL-MALONAMIDES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS CYTOVIA, INC. (US) 2005-04-28 WO disclosed