SCHEMBL624826

SCHEMBL624826

COc1ccc(-c2cnc3sc(N4CCOCC4)nn23)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 7/20 0.60
TP53 P04637 1/20 0.57
NPC1 O15118 1/20 0.55
MAPT P10636 1/20 0.55
RAB9A P51151 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
LMNA P02545 1/20 0.54
POLB P06746 1/20 0.54
THRB P10828 1/20 0.53
PIK3CA P42336 3/20 0.52
GAK O14976 4/20 0.49
KIT P10721 1/20 0.49
PIM1 P11309 1/20 0.49
FLT3 P36888 1/20 0.49
CDK7 P50613 1/20 0.49
KCNH2 Q12809 1/20 0.49
PIM3 Q86V86 1/20 0.49
HASPIN Q8TF76 1/20 0.49
PIM2 Q9P1W9 1/20 0.49
CFTR P13569 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624827 0.79 MAPT (0.62) TP53NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL1946275 0.79 FYN (0.69) FYNNPC1MAPTCFTR
SCHEMBL625796 0.77 PIK3CA (0.47) FYNTP53MAPTLMNAPOLB
SCHEMBL532633 0.77 PIK3CA (0.74) FYNLMNAPIK3CA
SCHEMBL2255821 0.77 FYN (0.78) FYNGAKHASPIN
SCHEMBL625391 0.76 HASPIN (0.52) FYNTP53MAPTLMNAPOLB
SCHEMBL18613295 0.75 FYN (1.00) FYNPIK3CAGAK
SCHEMBL27794654 0.74 FYN (0.73) FYNPIK3CA
SCHEMBL15975809 0.72 PIK3CA (0.77) FYNLMNAPIK3CA
SCHEMBL2255546 0.72 FYN (0.57) FYNPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed