SCHEMBL625391

SCHEMBL625391

COc1ncccc1-c1cnc2sc(N3CCOCC3)nn12

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HASPIN Q8TF76 9/20 0.52
KCNH2 Q12809 5/20 0.50
FLT3 P36888 3/20 0.48
CYP2C8 P10632 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2B6 P20813 1/20 0.48
CYP2C19 P33261 1/20 0.48
LMNA P02545 2/20 0.46
THRB P10828 2/20 0.46
KIT P10721 1/20 0.46
PIM1 P11309 1/20 0.46
CDK7 P50613 1/20 0.46
PIM3 Q86V86 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
MAPT P10636 1/20 0.44
POLB P06746 1/20 0.44
FYN P06241 1/20 0.43
TP53 P04637 2/20 0.43
CHEK1 O14757 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23244939 0.81 KCNH2 (0.76) HASPINKCNH2FLT3CYP2C8CYP2C9
SCHEMBL625392 0.80 F2RL3 (0.42) THRBMAPTCHEK1
SCHEMBL624826 0.76 FYN (0.60) HASPINKCNH2FLT3LMNATHRB
SCHEMBL626984 0.76 PIK3CA (0.48) HASPIN
SCHEMBL23245012 0.74 KCNH2 (0.62) HASPINKCNH2FLT3CYP2C8CYP2C9
SCHEMBL29695173 0.74 KCNH2 (0.62) HASPINKCNH2FLT3CYP2C8CYP2C9
SCHEMBL625796 0.71 PIK3CA (0.47) LMNATHRBMAPTPOLBFYN
SCHEMBL23288613 0.69 HASPIN (0.81) HASPINKCNH2FLT3CYP2C8CYP2C9
SCHEMBL624034 0.69 LMNA (0.48) LMNATHRBMAPTPOLBTP53
SCHEMBL27796786 0.68 SLC2A1 (0.46) CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed