SCHEMBL6249153

SCHEMBL6249153

CN1CCN(Cc2cccc(NC(=O)c3cc(NC(=O)c4ccnc(N5CCOCC5)c4)ccc3Cl)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.52
BTK Q06187 1/20 0.51
AURKA O14965 2/20 0.51
RPS6KB1 P23443 2/20 0.51
MAPK14 Q16539 8/20 0.49
MAPK13 O15264 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
KIT P10721 1/20 0.48
DDR1 Q08345 1/20 0.48
EGFR P00533 2/20 0.47
LMNA P02545 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KDM1A O60341 1/20 0.46
RCOR1 Q9UKL0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6251957 0.91 MAPK14 (0.56) AURKARPS6KB1MAPK14MAPK13KIT
SCHEMBL7855408 0.85 MAPK14 (0.64) MAPK14KITDDR1
SCHEMBL3938171 0.84 PPARG (0.61) PPARGMAPK14MAPK13L3MBTL1LMNA
SCHEMBL6968243 0.83 MAPK14 (0.61) MAPK14
SCHEMBL3932976 0.81 MAPK14 (0.60) PPARGMAPK14MAPK13L3MBTL1LMNA
SCHEMBL6980722 0.81 MAPK14 (0.65) MAPK14
SCHEMBL3938272 0.80 PPARG (0.59) PPARGMAPK14MAPK13LMNARAB9A
SCHEMBL5897072 0.80 MAPK14 (0.64) PPARGMAPK14MAPK13
SCHEMBL6253060 0.79 MAPK13 (0.61) PPARGMAPK14MAPK13LMNARAB9A
SCHEMBL6254089 0.79 MAPK13 (0.61) PPARGMAPK14MAPK13LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163212-B1 AMIDE DERIVATIVES ASTRAZENECA AB (SE) 2005-08-31 EP disclosed
US-6794380-B2 ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASE; ANTIALLERGENS ASTRAZENECA AB (SE) 2004-09-21 US disclosed
US-20030186966-A1 Amide derivatives ASTRAZENECA AB 2003-10-02 US disclosed
US-6548514-B1 Inhibitors of p38 kinase/cytokine suppressive binding protein (CSBP)/reactivating kinase (RK); 1-((pyridyl)aminocarbonyl)-3-((hetero)arylaminocarbonyl)benzene derivatives; treating cytokine related diseases and disorders ASTRAZENECA AB (SE) 2003-04-15 US disclosed
EP-1163212-A1 AMIDE DERIVATIVES AstraZeneca AB (SE) 2001-12-19 EP disclosed
WO-2000055120-A1 AMIDE DERIVATIVES ASTRAZENECA AB (SE) 2000-09-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030186966-A1 Amide derivatives IL6, IL6ST, IFNG PPARG 822/4885BTK 1602/4885AURKA 3240/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.