SCHEMBL624948

SCHEMBL624948

CCOc1cncc(-c2cn3nc(NCCCNC(=O)OC(C)(C)C)sc3n2)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 0.43
STK17B O94768 1/20 0.41
STK17A Q9UEE5 1/20 0.41
TTK P33981 1/20 0.40
PIK3CG P48736 1/20 0.40
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
DYRK1A Q13627 1/20 0.38
ACKR3 P25106 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624947 0.83 FYN (0.51) BRD4STK17BSTK17APIK3CG
SCHEMBL626774 0.82 PIK3CA (0.42) BRD4STK17BSTK17ATTKPIK3CG
SCHEMBL626603 0.77 STK17B (0.45) BRD4STK17BSTK17A
SCHEMBL625400 0.76 PIK3CA (0.43) PIK3CG
SCHEMBL625027 0.74 CA12 (0.42) STK17APIK3CGDYRK1A
SCHEMBL626663 0.71 BCHE (0.42) BRD4STK17BSTK17AACKR3
SCHEMBL626602 0.69 STK17B (0.47) BRD4STK17BSTK17AACKR3
SCHEMBL1945374 0.68 FYN (0.64) PIK3CGMAPTTP53
SCHEMBL1944741 0.68 FYN (0.47) PIK3CG
SCHEMBL15341063 0.66 STK17B (0.51) BRD4STK17BSTK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed