SCHEMBL626663

SCHEMBL626663

CC(C)(C)OC(=O)NCCNc1nn2cc(I)nc2s1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.42
BRD4 O60885 5/20 0.41
MALT1 Q9UDY8 1/20 0.38
ADORA3 P0DMS8 5/20 0.38
ADORA2A P29274 5/20 0.38
ADORA1 P30542 2/20 0.38
LATS1 O95835 1/20 0.37
STK17B O94768 1/20 0.37
STK17A Q9UEE5 1/20 0.37
SUV39H2 Q9H5I1 1/20 0.37
PI4KB Q9UBF8 1/20 0.36
ACKR3 P25106 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OGFRL1 Q5TC84 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626603 0.93 STK17B (0.45) BRD4ADORA3ADORA2AADORA1STK17B
SCHEMBL626662 0.77 ADORA3 (0.40) BCHEBRD4MALT1ADORA3ADORA2A
SCHEMBL626399 0.75 KDM1A (0.38)
SCHEMBL625400 0.75 PIK3CA (0.43) PI4KBPDE3BPDE3A
SCHEMBL626887 0.74 CKS1B (0.48) SUV39H2
SCHEMBL626211 0.72 IRAK1 (0.48) SUV39H2
SCHEMBL626602 0.71 STK17B (0.47) BRD4ADORA3ADORA2AADORA1STK17B
SCHEMBL1435757 0.70 PI4KB (0.46) BCHEBRD4MALT1LATS1STK17B
SCHEMBL627884 0.70 CCNA2 (0.50) ADORA2AACKR3
SCHEMBL760966 0.69 BCHE (0.53) BCHEBRD4MALT1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed