SCHEMBL626774

SCHEMBL626774

CC(C)(C)OC(=O)NCCCNc1nn2cc(-c3cnc(N)c(C(F)(F)F)c3)nc2s1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.42
STK17B O94768 1/20 0.42
STK17A Q9UEE5 1/20 0.42
CYP3A4 P08684 1/20 0.40
F2RL3 Q96RI0 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
P2RY14 Q15391 1/20 0.38
MAP3K12 Q12852 3/20 0.37
TTK P33981 1/20 0.37
BRD4 O60885 3/20 0.36
AAK1 Q2M2I8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625400 0.95 PIK3CA (0.43) PIK3CACYP3A4F2RL3PIK3CDPIK3CB
SCHEMBL626773 0.85 PIK3CA (0.51) PIK3CASTK17BSTK17ACYP3A4
SCHEMBL626145 0.83 F2RL3 (0.43) PIK3CACYP3A4F2RL3PIK3CDPIK3CB
SCHEMBL626625 0.83 PIK3CA (0.43) PIK3CACYP3A4F2RL3PIK3CDPIK3CB
SCHEMBL624948 0.82 BRD4 (0.43) STK17BSTK17APIK3CGTTKBRD4
SCHEMBL626299 0.81 PIK3CA (0.47) PIK3CACYP3A4F2RL3PIK3CDPIK3CB
SCHEMBL626269 0.81 F2RL3 (0.44) PIK3CACYP3A4F2RL3PIK3CDPIK3CB
SCHEMBL625399 0.80 PIK3CA (0.53) PIK3CACYP3A4
SCHEMBL626892 0.80 PIK3CA (0.42) PIK3CACYP3A4MAP3K12
SCHEMBL12474086 0.80 PIK3CA (0.47) PIK3CACYP3A4F2RL3PIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed