SCHEMBL6250997

SCHEMBL6250997

Nc1ccc2c3c(c4ccccc4cc13)C(=O)C=C2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 3/20 0.51
NQO1 P15559 1/20 0.42
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.36
KMT2A Q03164 3/20 0.36
LMNA P02545 2/20 0.36
HIF1A Q16665 2/20 0.36
MEN1 O00255 2/20 0.36
USP2 O75604 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
TP53 P04637 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
CDC25A P30304 3/20 0.35
CDC25C P30307 3/20 0.35
HSD17B10 Q99714 2/20 0.35
KEAP1 Q14145 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6250540 0.82 NQO1 (0.49) CES1NQO1ALDH1A1HPGDKMT2A
SCHEMBL6503129 0.78 CES1 (0.51) CES1NQO1ALDH1A1HPGDKMT2A
SCHEMBL29358751 0.78 CES1 (0.51) CES1NQO1ALDH1A1HPGDKMT2A
SCHEMBL5716919 0.71 CES1 (0.79) CES1NQO1ALDH1A1HPGDKMT2A
SCHEMBL4925761 0.70 ALDH1A1 (0.38) CES1ALDH1A1HPGDKMT2ALMNA
SCHEMBL716372 0.69 KMT2A (0.50) CES1ALDH1A1HPGDKMT2ALMNA
SCHEMBL7742191 0.69 CES1 (0.39) CES1ALDH1A1HPGDKMT2ALMNA
SCHEMBL380656 0.68 CES1 (1.00) CES1NQO1ALDH1A1HPGDKMT2A
SCHEMBL7213583 0.68 CES1 (0.72) CES1NQO1ALDH1A1HPGDKMT2A
SCHEMBL87570 0.67 CES1 (0.70) CES1NQO1ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE38723-E1 Haloalkyl derivatives of reporter molecules used to analyze metabolic activity in cells MOLECULAR PROBES, INC. (US) 2005-04-12 US disclosed
EP-0603266-A4 USE OF HALOALKYL DERIVATIVES OF REPORTER MOLECULES TO ANALYZE METABOLIC ACTIVITY IN CELLS. MOLECULAR PROBES INC (US) 1997-01-15 EP disclosed
EP-0603266-A1 USE OF HALOALKYL DERIVATIVES OF REPORTER MOLECULES TO ANALYZE METABOLIC ACTIVITY IN CELLS MOLECULAR PROBES, INC. (US) 1994-06-29 EP disclosed
WO-1993004192-A1 USE OF HALOALKYL DERIVATIVES OF REPORTER MOLECULES TO ANALYZE METABOLIC ACTIVITY IN CELLS MOLECULAR PROBES, INC. (US) 1993-03-04 WO disclosed