SCHEMBL626006

SCHEMBL626006

CCNC(=O)NC1CCCN(c2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)C1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.46
RIPK1 Q13546 1/20 0.41
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
KCNH2 Q12809 5/20 0.39
PIK3CD O00329 2/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
FLT3 P36888 1/20 0.36
HASPIN Q8TF76 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624865 0.90 PIK3CA (0.49) PIK3CARIPK1KCNH2PIK3CDPIK3CB
SCHEMBL626007 0.88 MAPT (0.51) PIK3CALMNATP53MAPTTHRB
SCHEMBL624869 0.84 PIK3CA (0.52) PIK3CARIPK1KCNH2PIK3CDPIK3CB
SCHEMBL625177 0.82 PIK3CA (0.49) PIK3CAKCNH2PIK3CDMAPTTHRB
SCHEMBL627329 0.82 PIK3CA (0.49) PIK3CAHASPIN
SCHEMBL627327 0.82 PIK3CA (0.49) PIK3CAHASPIN
SCHEMBL624633 0.81 PIK3CA (0.47) PIK3CALMNATP53KCNH2MAPT
SCHEMBL624990 0.81 PIK3CA (0.47) PIK3CARIPK1KCNH2
SCHEMBL625222 0.81 PIK3CA (0.48) PIK3CAKCNH2PIK3CDPIK3CBPIK3CG
SCHEMBL626391 0.81 PIK3CA (0.48) PIK3CAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed