SCHEMBL625189

SCHEMBL625189

CC(C)(C)OC(=O)NC(c1nn2c(-c3cnc(N)c(C(F)(F)F)c3)cnc2s1)C1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.46
MAP3K12 Q12852 7/20 0.36
RIPK1 Q13546 2/20 0.34
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626170 0.84 PIK3CA (0.53) PIK3CAMAP3K12
SCHEMBL625036 0.81 PIM1 (0.49)
SCHEMBL626700 0.81 PIK3CA (0.52) PIK3CAMAP3K12
SCHEMBL626888 0.79 AAK1 (0.34)
SCHEMBL625674 0.77 PIK3CA (0.50) PIK3CAMAP3K12
SCHEMBL626893 0.76 PIK3CA (0.49) PIK3CA
SCHEMBL626891 0.76 PIK3CA (0.49) PIK3CA
SCHEMBL625131 0.75 PIK3CA (0.49) PIK3CARIPK1
SCHEMBL625434 0.75 PIK3CA (0.50) PIK3CAMAP3K12
SCHEMBL624990 0.74 PIK3CA (0.47) PIK3CARIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed