SCHEMBL626888

SCHEMBL626888

CC(C)(C)OC(=O)NC(c1nn2c(I)cnc2s1)C1CCNCC1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.34
AKT1 P31749 2/20 0.34
SMYD3 Q9H7B4 3/20 0.32
PLAT P00750 1/20 0.32
GFER P55789 1/20 0.31
PTPRB P23467 1/20 0.31
TRPA1 O75762 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626212 0.89 AAK1 (0.33) AAK1AKT1JAK2JAK1
SCHEMBL625189 0.79 PIK3CA (0.46)
SCHEMBL625036 0.79 PIM1 (0.49)
SCHEMBL1585580 0.72 AAK1 (0.37) AAK1AKT1SMYD3TRPA1JAK2
SCHEMBL4116055 0.69 SMYD3 (0.53) AKT1SMYD3
SCHEMBL626398 0.69 FYN (0.44) JAK2JAK1
SCHEMBL627106 0.69 FYN (0.44) JAK2JAK1
SCHEMBL627316 0.69 FYN (0.34)
SCHEMBL6066440 0.69 AAK1 (0.44) AAK1AKT1SMYD3
SCHEMBL627225 0.69 CKS1B (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed