SCHEMBL625303

SCHEMBL625303

O=CC(c1ccccn1)C1(c2cccc(OC(F)(F)F)c2)CCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.43
TRPV3 Q8NET8 1/20 0.39
HDAC6 Q9UBN7 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
SLC6A9 P48067 1/20 0.36
CETP P11597 1/20 0.36
GRM5 P41594 1/20 0.35
SLC40A1 Q9NP59 1/20 0.34
TACR1 P25103 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
PKLR P30613 1/20 0.33
OPRL1 P41146 1/20 0.33
SCN9A Q15858 2/20 0.33
PDE2A O00408 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625892 0.84 TRPV3 (0.41) TRPV3HDAC6HDAC3HDAC1HDAC2
SCHEMBL624452 0.84 NR1I2 (0.59) NR1I2TRPV3HDAC6HDAC3HDAC1
SCHEMBL626252 0.82 TRPV3 (0.44) TRPV3HDAC6HDAC3HDAC1HDAC2
SCHEMBL625907 0.81 NR1I2 (0.46) NR1I2TRPV3HDAC6HDAC3HDAC1
SCHEMBL14893798 0.75 NR1I2 (0.57) NR1I2TRPV3HDAC6HDAC3HDAC1
SCHEMBL14894470 0.75 NR1I2 (0.57) NR1I2TRPV3HDAC6HDAC3HDAC1
SCHEMBL14893800 0.75 NR1I2 (0.57) NR1I2TRPV3HDAC6HDAC3HDAC1
SCHEMBL624777 0.75 NR1I2 (0.43) NR1I2TRPV3HDAC6HDAC3HDAC1
SCHEMBL625410 0.75 TRPV3 (0.68) TRPV3SLC6A2SLC6A4SLC6A3
SCHEMBL625906 0.74 NR1I2 (0.46) NR1I2TRPV3HDAC6HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2603490-A1 NOVEL TRPV3 MODULATORS AbbVie Inc. (US) 2013-06-19 EP disclosed
WO-2012019315-A1 NOVEL TRPV3 MODULATORS ABBOTT LABORATORIES (US) 2012-02-16 WO disclosed