SCHEMBL625348

SCHEMBL625348

O=C1CCNC(=Cc2ccc(Br)cc2)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
PIM1 P11309 1/20 0.44
PIM2 Q9P1W9 1/20 0.44
MEN1 O00255 1/20 0.40
CISD1 Q9NZ45 1/20 0.40
TDP1 Q9NUW8 1/20 0.37
PARP10 Q53GL7 2/20 0.36
PARP11 Q9NR21 1/20 0.36
PARP1 P09874 1/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
ALPL P05186 1/20 0.35
ALPI P09923 1/20 0.35
ALOX15 P16050 1/20 0.35
PTGS2 P35354 1/20 0.35
MAPT P10636 2/20 0.35
EGFR P00533 1/20 0.35
XDH P47989 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625347 1.00 KMT2A (0.45) KMT2AMAOAMAOBPIM1PIM2
SCHEMBL28371952 1.00 KMT2A (0.45) KMT2AMAOAMAOBPIM1PIM2
SCHEMBL28885464 0.83 PIM1 (0.44) MAOAMAOBPIM1PIM2PARP10
SCHEMBL28927253 0.83 PARP10 (0.33) PARP10PARP11PARP1
SCHEMBL28885466 0.83 PIM1 (0.44) MAOAMAOBPIM1PIM2PARP10
SCHEMBL625684 0.83 CYP2C9 (0.47) KMT2AMAOAMAOBMEN1TDP1
SCHEMBL625683 0.83 CYP2C9 (0.47) KMT2AMAOAMAOBMEN1TDP1
SCHEMBL624212 0.83 HSD11B1 (0.47) KMT2AMAOAMAOBPIM1PIM2
SCHEMBL624211 0.83 HSD11B1 (0.47) KMT2AMAOAMAOBPIM1PIM2
SCHEMBL28375460 0.83 HSD11B1 (0.47) KMT2AMAOAMAOBPIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110878095-B Curcumin bifunctional molecule and preparation method and application thereof 中山大学 2023-01-24 CN disclosed
CN-115232068-A Compound and preparation method and application thereof 北京中医药大学 2022-10-25 CN disclosed
CN-110878095-A Curcumin bifunctional molecule and preparation method and application thereof 中山大学 2020-03-13 CN disclosed
WO-2012021692-A1 CURCUMIN ANALOGS AND METHODS OF USE THEREOF RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2012-02-16 WO disclosed