SCHEMBL625512

SCHEMBL625512

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1nn3cc(-c4cccc(OC(F)(F)F)c4)nc3s1)CC2

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
THRB P10828 3/20 0.44
MAPT P10636 13/20 0.43
RXFP1 Q9HBX9 1/20 0.40
F2RL3 Q96RI0 2/20 0.39
CYP11B2 P19099 1/20 0.39
SCD5 Q86SK9 1/20 0.38
PIM1 P11309 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623996 0.95 THRB (0.42) THRBMAPTRXFP1F2RL3CYP11B2
SCHEMBL624528 0.92 CYP3A4 (0.41) THRBMAPTRXFP1CYP11B2SCD5
SCHEMBL625496 0.86 PIM1 (0.39) THRBMAPTF2RL3SCD5PIM1
SCHEMBL625742 0.85 THRB (0.43) THRBMAPTRXFP1F2RL3PIM1
SCHEMBL625511 0.85 PIM1 (0.45) PIM1
SCHEMBL623949 0.84 PIM1 (0.47) THRBMAPTRXFP1F2RL3PIM1
SCHEMBL624454 0.82 PIM1 (0.45) F2RL3PIM1
SCHEMBL625255 0.82 PIM3 (0.48) THRBMAPTRXFP1F2RL3PIM1
SCHEMBL624740 0.81 PIM1 (0.48) THRBMAPTRXFP1F2RL3PIM1
SCHEMBL623995 0.80 PIM1 (0.44) CYP11B2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed