SCHEMBL623996

SCHEMBL623996

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1nn3cc(-c4cccc(OC(F)(F)F)c4)nc3s1)C2

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
THRB P10828 3/20 0.42
MAPT P10636 10/20 0.41
CYP11B2 P19099 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
SCD5 Q86SK9 1/20 0.39
F2RL3 Q96RI0 2/20 0.38
RET P07949 1/20 0.38
PIM1 P11309 1/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
MGLL Q99685 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624528 0.96 CYP3A4 (0.41) THRBMAPTCYP11B2RXFP1SCD5
SCHEMBL625512 0.95 THRB (0.44) THRBMAPTCYP11B2RXFP1SCD5
SCHEMBL623995 0.85 PIM1 (0.44) CYP11B2RETPIM1
SCHEMBL623207 0.85 PIM1 (0.48) THRBMAPTRXFP1F2RL3PIM1
SCHEMBL625496 0.84 PIM1 (0.39) THRBMAPTSCD5F2RL3PIM1
SCHEMBL625742 0.84 THRB (0.43) THRBMAPTRXFP1F2RL3PIM1
SCHEMBL624527 0.82 PIM1 (0.43) RETPIM1
SCHEMBL624454 0.81 PIM1 (0.45) F2RL3RETPIM1
SCHEMBL625511 0.80 PIM1 (0.45) PIM1
SCHEMBL623949 0.80 PIM1 (0.47) THRBMAPTRXFP1F2RL3PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed