SCHEMBL625511

SCHEMBL625511

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1nn3c(-c4cccc(OC(F)(F)F)c4)cnc3s1)CC2

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 11/20 0.45
DYRK1A Q13627 6/20 0.44
KCNH2 Q12809 1/20 0.42
FYN P06241 1/20 0.42
HASPIN Q8TF76 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623995 0.95 PIM1 (0.44) PIM1DYRK1AKCNH2FYNHASPIN
SCHEMBL624527 0.92 PIM1 (0.43) PIM1DYRK1AKCNH2
SCHEMBL625495 0.85 PIM1 (0.46) PIM1KCNH2FYNHASPIN
SCHEMBL625741 0.85 PIM1 (0.45) PIM1DYRK1AFYN
SCHEMBL625512 0.85 THRB (0.44) PIM1
SCHEMBL623948 0.85 DYRK1A (0.47) PIM1DYRK1AKCNH2HASPIN
SCHEMBL624453 0.82 PIM1 (0.51) PIM1KCNH2FYNHASPIN
SCHEMBL625254 0.81 PIM3 (0.51) PIM1DYRK1AKCNH2HASPIN
SCHEMBL624739 0.81 PIM1 (0.47) PIM1DYRK1AKCNH2HASPIN
SCHEMBL623996 0.80 THRB (0.42) PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed