SCHEMBL6257167

SCHEMBL6257167

CN(C)C(CC=CC=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
OPRM1 P35372 2/20 0.40
OPRD1 P41143 1/20 0.40
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HTR2A P28223 2/20 0.37
HRH1 P35367 2/20 0.37
OPRK1 P41145 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
KAT2B Q92831 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3825964 0.82 CHRNB2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1
SCHEMBL27759532 0.79 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1
SCHEMBL28501662 0.79 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1
SCHEMBL4755637 0.77 LMNA (0.41) ALDH1A1KDM4EL3MBTL1HTR2AHRH1
SCHEMBL10454477 0.77 TAAR1 (0.45) ALDH1A1LMNATRPA1ALOX5MAPK1
SCHEMBL173965 0.74 SMN1; SMN2 (0.49) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1
Iodide SCHEMBL29054398 0.73 SMN1; SMN2 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1
SCHEMBL10372161 0.73 KDM4E (0.48) KDM4EL3MBTL1CYP2D6CYP2C19LMNA
Bromide SCHEMBL1980740 0.73 SMN1; SMN2 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1
Water SCHEMBL2110704 0.73 SMN1; SMN2 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1524262-A1 Inhibitors of histone deacetylase Methylgene, Inc. (CA) 2005-04-20 EP disclosed