SCHEMBL625732

SCHEMBL625732

CS(=O)(=O)NC1CCN(c2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)C1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.53
KCNH2 Q12809 4/20 0.41
MAP3K12 Q12852 1/20 0.39
AKT1 P31749 2/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
TNF P01375 1/20 0.35
PDE2A O00408 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624869 0.95 PIK3CA (0.52) PIK3CAKCNH2MAP3K12PIK3CDPIK3CB
SCHEMBL624967 0.95 PIK3CA (0.55) PIK3CAKCNH2MAP3K12
SCHEMBL625733 0.87 MAP3K12 (0.42) PIK3CAMAP3K12
SCHEMBL626168 0.84 PIK3CA (0.53) PIK3CAKCNH2MAP3K12
SCHEMBL624990 0.84 PIK3CA (0.47) PIK3CAKCNH2
SCHEMBL625432 0.83 PIK3CA (0.50) PIK3CAKCNH2MAP3K12PIK3CDPIK3CB
SCHEMBL625227 0.83 PIK3CA (0.55) PIK3CAKCNH2MAP3K12
SCHEMBL624865 0.82 PIK3CA (0.49) PIK3CAKCNH2PIK3CDPIK3CBPIK3CG
SCHEMBL624870 0.82 MAPT (0.42) PIK3CAMAP3K12
SCHEMBL626619 0.81 PIK3CA (0.55) PIK3CAKCNH2MAP3K12TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed