SCHEMBL625859

SCHEMBL625859

CC(C)(C)OC(=O)N1CCN(c2ncc(-c3cnc4sc(N(C5CCNCC5)S(C)(=O)=O)nn34)cc2C(F)(F)F)CC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.43
GPR119 Q8TDV5 8/20 0.35
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
KIT P10721 2/20 0.34
ALK Q9UM73 2/20 0.33
RIPK1 Q13546 1/20 0.33
RET P07949 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625860 0.79 GPR119 (0.47) PIK3CAGPR119RIPK1
SCHEMBL2121133 0.74 PIK3CA (0.77) PIK3CAALK
SCHEMBL624921 0.74 PIK3CA (0.49) PIK3CAGPR119RIPK1
SCHEMBL625421 0.72 PIK3CA (0.52) PIK3CAGPR119KITRIPK1
SCHEMBL624393 0.71 FYN (0.46) PIK3CA
SCHEMBL625127 0.69 PIK3CA (0.48) PIK3CARIPK1
SCHEMBL29029902 0.69 DDB1 (0.45) GPR119KITALK
SCHEMBL625653 0.69 PIK3CA (0.54) PIK3CA
SCHEMBL31410416 0.68 KMT2A (0.57) GPR119KIT
SCHEMBL31410432 0.68 KMT2A (0.57) GPR119KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed