SCHEMBL625910

SCHEMBL625910

CC(C)C(NC(=O)OCc1ccccc1)C(=O)NC(CC(=O)OC(C)(C)C)C(O)COc1c(F)c(F)cc(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSD P07339 2/20 0.44
CASP3 P42574 8/20 0.44
CASP6 P55212 7/20 0.44
CASP8 Q14790 7/20 0.44
REN P00797 4/20 0.43
KLK5 Q9Y337 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4434235 1.00 CTSD (0.44) CTSDCASP3CASP6CASP8REN
SCHEMBL10073352 1.00 CTSD (0.44) CTSDCASP3CASP6CASP8REN
SCHEMBL17261863 0.92 REN (0.43) CASP3CASP6CASP8RENKLK5
SCHEMBL79910 0.92 SYK (0.44) KLK5
SCHEMBL3213032 0.92 SYK (0.44) KLK5
SCHEMBL79132 0.92 SYK (0.44) KLK5
SCHEMBL14598451 0.86 REN (0.40) CTSDCASP3CASP6CASP8REN
SCHEMBL626605 0.85 CASP3 (0.51) CASP3CASP6CASP8
SCHEMBL10073348 0.85 CASP3 (0.60) CASP3CASP6CASP8
SCHEMBL626915 0.85 CASP3 (0.60) CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021800-A2 CASPASE INHIBITORS AS THERAPEUTICS FOR NEURAL AND ORGAN INJURY AND IMAGING BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed