SCHEMBL6259170

SCHEMBL6259170

NC(=O)c1cn(-c2ccccc2)nc1-c1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.75
CA1 P00915 5/20 0.75
CA2 P00918 5/20 0.75
CA9 Q16790 5/20 0.75
MAPT P10636 1/20 0.67
AURKA O14965 3/20 0.65
TP53 P04637 1/20 0.65
ALDH1A1 P00352 7/20 0.64
KDM4E B2RXH2 4/20 0.64
L3MBTL1 Q9Y468 2/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
HPGD P15428 1/20 0.64
HSD17B10 Q99714 1/20 0.64
PKM P14618 1/20 0.63
ATM Q13315 1/20 0.58
KDM5B Q9UGL1 1/20 0.58
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
LMNA P02545 1/20 0.58
GAA P10253 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18292676 0.87 KMT2A (0.64) CA12CA1CA2CA9MAPT
SCHEMBL4501557 0.87 ALDH1A1 (0.82) CA12CA1CA2CA9MAPT
SCHEMBL23928504 0.85 CA12 (0.75) CA12CA1CA2CA9MAPT
SCHEMBL6686483 0.84 CA12 (0.57) CA12CA1CA2CA9MAPT
Propionic Acid SCHEMBL28500081 0.84 CA12 (0.64) CA12CA1CA2CA9MAPT
SCHEMBL5812722 0.84 MAPT (0.67) CA12CA1CA2CA9MAPT
SCHEMBL28771391 0.84 ALDH1A1 (0.78) MAPTAURKATP53ALDH1A1KDM4E
SCHEMBL4498839 0.81 MAPT (0.63) CA12CA1CA2CA9MAPT
SCHEMBL976547 0.81 AURKA (0.74) CA12CA9MAPTAURKATP53
SCHEMBL16597905 0.80 CA12 (0.59) CA12CA1CA2CA9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005061462-A2 DIARYL PYRAZOLE DERIVATIVES AND THEIR USE AS NEUROKININ-3 RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2005-07-07 WO disclosed