SCHEMBL6260698

SCHEMBL6260698

COc1ccccc1C1(C(Cl)C=O)CCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.40
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
HTT P42858 1/20 0.34
HPGD P15428 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LPAR1 Q92633 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CHRM2 P08172 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6259081 0.79 SIGMAR1 (0.43) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL13107316 0.77 SIGMAR1 (0.43) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL13107313 0.77 SIGMAR1 (0.43) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL3443490 0.77 SIGMAR1 (0.43) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL7570645 0.74 HDAC4 (0.43) OPRM1OPRD1OPRK1OPRL1PSEN1
SCHEMBL7564524 0.73 PSEN1 (0.43) OPRM1OPRD1OPRK1OPRL1PSEN1
SCHEMBL4445384 0.73 HDAC4 (0.40) OPRM1OPRK1KMT2AALDH1A1HDAC3
SCHEMBL14388188 0.71 SIGMAR1 (0.41) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL30040141 0.70 APP (0.46) SIGMAR1KMT2AHTTALDH1A1LPAR1
SCHEMBL21034069 0.70 APP (0.46) SIGMAR1KMT2AHTTALDH1A1LPAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005077463-A2 LIGAND FOR A MONOAMINE RECEPTOR OR TRANSPORTER FOR TREATING ADDICTION OR DEPENDENCE SEPRACOR INC. (US) 2005-08-25 WO disclosed
EP-1318988-A2 LIGANDS FOR MONOAMINE RECEPTORS AND TRANSPORTERS, AND METHODS OF USE THEREOF (NEUROTRANSMISSION) Sepracor, Inc. (US) 2003-06-18 EP disclosed
WO-2002022572-A2 LIGANDS FOR MONOAMINE RECEPTORS AND TRANSPORTERS, AND METHODS OF USE THEREOF (NEUROTRANSMISSION) SEPRACOR, INC. (US) 2002-03-21 WO disclosed