SCHEMBL626108

SCHEMBL626108

Nc1ncc(-c2cn3nc(NC4CC5(CCNCC5)C4)sc3n2)cc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 19/20 0.42
DLK1 P80370 1/20 0.40
PIK3CA P42336 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625236 0.88 MAP3K12 (0.45) MAP3K12DLK1PIK3CA
SCHEMBL626107 0.84 PIK3CA (0.48) PIK3CA
SCHEMBL625408 0.83 MAP4K1 (0.39) MAP3K12DLK1PIK3CA
SCHEMBL625459 0.82 MAP3K12 (0.41) MAP3K12DLK1PIK3CA
SCHEMBL625636 0.82 MAP3K12 (0.44) MAP3K12DLK1PIK3CA
SCHEMBL624439 0.81 MAP3K12 (0.41) MAP3K12DLK1PIK3CA
SCHEMBL627440 0.81 FYN (0.45) MAP3K12DLK1PIK3CA
SCHEMBL625468 0.81 MAP3K12 (0.42) MAP3K12DLK1PIK3CA
SCHEMBL625549 0.81 F2RL3 (0.51)
SCHEMBL625301 0.80 MAP3K12 (0.44) MAP3K12DLK1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed