SCHEMBL625408

SCHEMBL625408

CC(C)(C)OC(=O)N1CCC2(CC1)CC(Nc1nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s1)C2

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 1/20 0.39
MAP3K12 Q12852 13/20 0.39
PIK3CA P42336 2/20 0.39
DLK1 P80370 1/20 0.38
SYK P43405 1/20 0.38
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
RORC P51449 1/20 0.37
NAMPT P43490 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625128 0.90 CCNA2 (0.46) MAP4K1MAP3K12PIK3CASYKCCNA2
SCHEMBL625407 0.87 PIK3CA (0.45) PIK3CANAMPT
SCHEMBL627432 0.86 RET (0.40) MAP4K1MAP3K12PIK3CADLK1
SCHEMBL627020 0.85 RET (0.40) MAP3K12PIK3CA
SCHEMBL623829 0.84 F2RL3 (0.48) SYKNAMPT
SCHEMBL625456 0.83 MAP3K12 (0.41) MAP4K1MAP3K12PIK3CASYKCCNA2
SCHEMBL625422 0.83 PIK3CA (0.42) MAP3K12PIK3CA
SCHEMBL626108 0.83 MAP3K12 (0.42) MAP3K12PIK3CADLK1
SCHEMBL626123 0.82 RET (0.43) MAP3K12PIK3CA
SCHEMBL624985 0.82 KDM4E (0.40) MAP4K1MAP3K12PIK3CASYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed