SCHEMBL626579

SCHEMBL626579

NCCC(N)c1nn2c(-c3cnc(N)c(C(F)(F)F)c3)cnc2s1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.56
MAP3K12 Q12852 10/20 0.38
TNF P01375 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626580 0.82 PIK3CA (0.45) PIK3CAMAP3K12
SCHEMBL626700 0.79 PIK3CA (0.52) PIK3CAMAP3K12
SCHEMBL626268 0.78 PIK3CA (0.59) PIK3CA
SCHEMBL626144 0.77 PIK3CA (0.57) PIK3CA
SCHEMBL624388 0.73 PIK3CA (0.55) PIK3CAMAP3K12
SCHEMBL12474083 0.72 PIK3CA (0.57) PIK3CA
SCHEMBL624411 0.72 PIK3CA (0.54) PIK3CA
SCHEMBL532031 0.72 PIK3CA (1.00) PIK3CATNF
SCHEMBL625201 0.72 PIK3CA (0.48) PIK3CAMAP3K12
SCHEMBL15975831 0.71 PIK3CA (0.73) PIK3CATNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed