SCHEMBL626580

SCHEMBL626580

NCCC(N)c1nn2cc(-c3cnc(N)c(C(F)(F)F)c3)nc2s1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.45
MAP3K12 Q12852 16/20 0.45
F2RL3 Q96RI0 1/20 0.43
DLK1 P80370 1/20 0.42
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626579 0.82 PIK3CA (0.56) PIK3CAMAP3K12
SCHEMBL626269 0.80 F2RL3 (0.44) PIK3CAMAP3K12F2RL3
SCHEMBL626145 0.78 F2RL3 (0.43) PIK3CAMAP3K12F2RL3
SCHEMBL624389 0.75 MAP3K12 (0.43) PIK3CAMAP3K12F2RL3DLK1
SCHEMBL12474086 0.74 PIK3CA (0.47) PIK3CAMAP3K12F2RL3
SCHEMBL624412 0.74 MAP3K12 (0.45) PIK3CAMAP3K12MAPT
SCHEMBL532032 0.74 PIK3CA (0.68) PIK3CAMAP3K12F2RL3TP53MAPT
SCHEMBL532091 0.73 PIK3CA (0.71) PIK3CAMAP3K12F2RL3
SCHEMBL625202 0.73 MAP3K12 (0.43) MAP3K12TP53MAPT
SCHEMBL533618 0.73 PIK3CA (0.51) PIK3CAMAP3K12F2RL3TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed