SCHEMBL626662

SCHEMBL626662

CC(C)(C)OC(=O)NCCNc1nn2c(I)cnc2s1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.40
ADORA2A P29274 5/20 0.40
BCHE P06276 1/20 0.39
STK17B O94768 1/20 0.39
STK17A Q9UEE5 1/20 0.39
BRD4 O60885 2/20 0.39
MALT1 Q9UDY8 1/20 0.38
CSNK1D P48730 1/20 0.38
ACKR3 P25106 2/20 0.38
ADORA1 P30542 2/20 0.38
LATS1 O95835 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GFER P55789 1/20 0.37
FYN P06241 3/20 0.36
FPR3 P25089 2/20 0.36
FPR2 P25090 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626602 0.93 STK17B (0.47) ADORA3ADORA2ASTK17BSTK17ABRD4
SCHEMBL626663 0.77 BCHE (0.42) ADORA3ADORA2ABCHESTK17BSTK17A
SCHEMBL25810293 0.76 BCHE (0.42) ADORA3ADORA2ABCHESTK17BSTK17A
SCHEMBL1650182 0.76 ALPL (0.46) ACKR3FYN
SCHEMBL625399 0.76 PIK3CA (0.53) CSNK1DFYN
SCHEMBL626398 0.75 FYN (0.44) FYN
SCHEMBL627066 0.74 KDM4E (0.46) ACKR3FYN
SCHEMBL626886 0.74 CKS1B (0.50)
SCHEMBL25003064 0.73 STK17B (0.49) BCHESTK17BSTK17ABRD4MALT1
SCHEMBL23244988 0.73 KCNH2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed