SCHEMBL626701

SCHEMBL626701

Nc1ncc(-c2cnc3sc(NCC4CCNCC4)nn23)cc1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.52
PIK3CA P42336 9/20 0.52
FYN P06241 8/20 0.52
PIM1 P11309 2/20 0.42
KIT P10721 1/20 0.39
FLT3 P36888 1/20 0.39
CDK7 P50613 1/20 0.39
KCNH2 Q12809 1/20 0.39
PIM3 Q86V86 1/20 0.39
HASPIN Q8TF76 1/20 0.39
PIM2 Q9P1W9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627612 0.89 FYN (0.56) MKNK1PIK3CAFYN
SCHEMBL627610 0.89 FYN (0.56) MKNK1PIK3CAFYN
SCHEMBL625672 0.88 PIK3CA (0.53) MKNK1PIK3CAFYN
SCHEMBL627782 0.87 PIK3CA (0.56) MKNK1PIK3CAFYNPIM1KIT
SCHEMBL625235 0.86 FYN (0.52) PIK3CAFYNHASPIN
SCHEMBL626581 0.84 FYN (0.47) MKNK1PIK3CAFYN
SCHEMBL626702 0.84 MAP3K12 (0.43) PIK3CAFLT3
SCHEMBL626288 0.83 PIK3CA (0.51) PIK3CAFYNPIM1KITFLT3
SCHEMBL625674 0.82 PIK3CA (0.50) PIK3CAFYN
SCHEMBL624984 0.82 PIK3CA (0.48) MKNK1PIK3CAFYNPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed