SCHEMBL627782

SCHEMBL627782

CO[C@H]1CC[C@H](CNc2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)CC1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.56
MKNK1 Q9BUB5 1/20 0.52
FYN P06241 8/20 0.52
HASPIN Q8TF76 2/20 0.41
KIT P10721 1/20 0.40
PIM1 P11309 1/20 0.40
FLT3 P36888 1/20 0.40
CDK7 P50613 1/20 0.40
KCNH2 Q12809 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627610 0.89 FYN (0.56) PIK3CAMKNK1FYN
SCHEMBL627612 0.89 FYN (0.56) PIK3CAMKNK1FYN
SCHEMBL625672 0.88 PIK3CA (0.53) PIK3CAMKNK1FYN
SCHEMBL626701 0.87 MKNK1 (0.52) PIK3CAMKNK1FYNHASPINKIT
SCHEMBL624984 0.83 PIK3CA (0.48) PIK3CAMKNK1FYNPIM1
SCHEMBL626581 0.82 FYN (0.47) PIK3CAMKNK1FYN
SCHEMBL627785 0.81 PIK3CA (0.56) PIK3CAPIM1
SCHEMBL627784 0.81 PIK3CA (0.56) PIK3CAPIM1
SCHEMBL627372 0.80 PIK3CA (0.57) PIK3CAHASPINKITPIM1FLT3
SCHEMBL626268 0.79 PIK3CA (0.59) PIK3CAMKNK1FYNHASPINKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed