SCHEMBL624984

SCHEMBL624984

CC(C)(C)OC(=O)N1CCC(CNc2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)CC1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.48
FYN P06241 7/20 0.47
MKNK1 Q9BUB5 1/20 0.44
RIPK1 Q13546 2/20 0.42
PIM1 P11309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625127 0.88 PIK3CA (0.48) PIK3CAFYNRIPK1
SCHEMBL626581 0.87 FYN (0.47) PIK3CAFYNMKNK1
SCHEMBL624985 0.86 KDM4E (0.40) PIK3CA
SCHEMBL625672 0.86 PIK3CA (0.53) PIK3CAFYNMKNK1
SCHEMBL626544 0.86 ACKR3 (0.55) PIK3CAFYNRIPK1
SCHEMBL624920 0.84 PIK3CA (0.46) PIK3CARIPK1
SCHEMBL627782 0.83 PIK3CA (0.56) PIK3CAFYNMKNK1PIM1
SCHEMBL628028 0.83 FYN (0.56) FYNMKNK1PIM1
SCHEMBL627612 0.83 FYN (0.56) PIK3CAFYNMKNK1
SCHEMBL627610 0.83 FYN (0.56) PIK3CAFYNMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed