SCHEMBL626773

SCHEMBL626773

CC(C)(C)OC(=O)NCCCNc1nn2c(-c3cnc(N)c(C(F)(F)F)c3)cnc2s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.51
FYN P06241 5/20 0.43
STK17B O94768 1/20 0.41
STK17A Q9UEE5 1/20 0.41
KIT P10721 1/20 0.41
PIM1 P11309 1/20 0.41
FLT3 P36888 1/20 0.41
CDK7 P50613 1/20 0.41
KCNH2 Q12809 1/20 0.41
PIM3 Q86V86 1/20 0.41
HASPIN Q8TF76 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
CYP3A4 P08684 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
CSNK2A2 P19784 1/20 0.38
CSNK2A1 P68400 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625399 0.95 PIK3CA (0.53) PIK3CAFYNKITPIM1FLT3
SCHEMBL626774 0.85 PIK3CA (0.42) PIK3CASTK17BSTK17ACYP3A4
SCHEMBL626144 0.83 PIK3CA (0.57) PIK3CAFYNKITPIM1FLT3
SCHEMBL626544 0.81 ACKR3 (0.55) PIK3CAFYN
SCHEMBL626298 0.81 PIK3CA (0.53) PIK3CAFYNKITPIM1FLT3
SCHEMBL626268 0.81 PIK3CA (0.59) PIK3CAFYNKITPIM1FLT3
SCHEMBL624947 0.80 FYN (0.51) FYNSTK17BSTK17A
SCHEMBL625400 0.80 PIK3CA (0.43) PIK3CACYP3A4PDE3BPDE3A
SCHEMBL626893 0.79 PIK3CA (0.49) PIK3CAFYNHASPIN
SCHEMBL626891 0.79 PIK3CA (0.49) PIK3CAFYNHASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed