SCHEMBL626544

SCHEMBL626544

CC(C)(C)OC(=O)N1CCN(CCNc2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)CC1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 7/20 0.55
PIK3CA P42336 10/20 0.48
FYN P06241 2/20 0.44
RIPK1 Q13546 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624984 0.86 PIK3CA (0.48) PIK3CAFYNRIPK1
SCHEMBL625127 0.85 PIK3CA (0.48) PIK3CAFYNRIPK1
SCHEMBL625399 0.83 PIK3CA (0.53) PIK3CAFYN
SCHEMBL626288 0.83 PIK3CA (0.51) PIK3CAFYN
SCHEMBL625421 0.82 PIK3CA (0.52) PIK3CARIPK1
SCHEMBL625407 0.81 PIK3CA (0.45) PIK3CAFYNRIPK1
SCHEMBL626773 0.81 PIK3CA (0.51) PIK3CAFYN
SCHEMBL623028 0.81 ACKR3 (0.54) ACKR3FYN
SCHEMBL624920 0.80 PIK3CA (0.46) PIK3CARIPK1
SCHEMBL627014 0.79 ACKR3 (0.63) ACKR3FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed